No.97 文献リスト [GPCR PathHunter Arrestin]-6 新規追加

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文献リスト [GPCR PathHunter Arrestin]-1
文献リスト [GPCR PathHunter Arrestin]-2
文献リスト [GPCR PathHunter Arrestin]-3
文献リスト [GPCR PathHunter Arrestin]-4
文献リスト [GPCR PathHunter Arrestin]-5

GPCR Target	Reference
ADRB1	Rastogi T, Leder C, Kummerer K. (2015). Re-Designing of Existing Pharmaceuticals for Environmental Biodegradability: A tiered approach with β-Blocker Propranolol as an example. Environ Sci Technol. [Epub ahead of print]
CNR2	Mukhopadhyay P, Baggelaar M, Erdelyi K, Cao Z, Cinar R, Fezza F, Ignatowska-Jankowska B, Wilkerson J, van Gils N, Hansen T, Ruben M, Soethoudt M, Heitman L, Kunos G, Maccarrone M, Lichtman A, Pacher P, van der Stelt M. (2015). The novel, orally available and peripherally restricted selective cannabinoid CB2 -receptor agonist LEI-101 prevents cisplatin-induced nephrotoxicity. Br J Pharmacol.[Epub ahead of print]
GPR18	Chiang N, Dalli J, Colas RA, Serhan CN. (2015) Identification of resolvin D2 receptor mediating resolution of infections and organ protection. J Exp Med. [Epub ahead of print]
GLP1R	Nakane A, Gotoh Y, Ichihara J, Nagata H. (2015). New Screening Strategy and Analysis for Identification of Allosteric Modulators for GLP-1 Receptor Using GLP-1(9-36)amide. Anal Biochem [Epub ahead of print]
S1P1 (EDG1)	Taylor SJ, Demont EH, Gray J, Deeks N, Patel A, Nguyen D, Taylor M, Hood S, Watson R, Bit RA, McClure F, Ashall H, Witherington J (2015). Navigating CYP1A induction and arylhydrocarbon receptor agonism in drug discovery. A case history with S1P1 agonists. J Med Chem [Epub ahead of print]
OPRM1	Bisignano P, Burford NT, Shang Y, Marlow B, Livingston K, Fenton AM, Rockwell K, Budenholzer L, Traynor JR, Gerritz SW, Alt A, Filizola M. (2015). Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the mu-Opioid Receptor. J Chem Inf Model [Epub ahead of print]
PAR1	Hawes BE, Zhai Y, Hesk D, Wirth M, Wei H, Chintala M, Seiffert D. (2015). In vitro pharmacological characterization of vorapaxar, a novel platelet thrombin receptor antagonist. Eur J Pharmacol. [Epub ahead of print]

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